Uses

What is betaxolol used for?

Betaxolol is commonly used to lower high blood pressure (hypertension).

Betaxolol may also be used for other conditions as determined by your healthcare provider.

How does betaxolol work (mechanism of action)?

Betaxolol blocks beta-1 receptors in your heart. These receptors normally bind to hormones called catecholamines. When catecholamines bind to these receptors, it causes your heart to beat harder and faster. Blocking these receptors helps your heart beat more slowly. These effects can help lower blood pressure, and may reduce your risk for heart attack and stroke. 

How is betaxolol supplied (dosage forms)?

Betaxolol is available in the following dosage forms that are taken by mouth.

  • 10 mg oral tablets
  • 20 mg oral tablets

How should I store betaxolol?

Betaxolol should be stored at room temperature, between 68 F to 77 F (20 C to 25 C). It can be exposed to temperatures between 59 F to 86 F (15 C to 30 C), for shorter periods of time, such as when transporting it. Store in a cool, dry place.

Side Effects

What are the most common side effects of betaxolol?

The most common side effects of betaxolol are listed below. Tell your healthcare provider if you have any of these side effects that bother you.

  • Tiredness
  • Dizziness
  • Headache
  • Slow heartbeat

There may be other side effects of betaxolol that are not listed here. Contact your healthcare provider if you think you are having a side effect of a medicine. In the U.S., you can report side effects to the FDA at www.fda.gov/medwatch or by calling 800-FDA-1088. In Canada, you can report side effects to Health Canada at www.health.gc.ca/medeffect or by calling 866-234-2345.

What are the serious side effects of betaxolol?

While less common, the most serious side effects of betaxolol are described below, along with what to do if they happen.

New or Worsening Heart Failure. Betaxolol may worsen existing heart failure or cause fluid buildup in your body. For individuals with underlying heart disease or heart damage, betaxolol can potentially lead to heart failure over time. Tell your healthcare provider right away if you have any of the following symptoms.

  • Shortness of breath or trouble breathing, especially while lying down
  • Swelling in your feet, ankles, or legs
  • Unusually fast weight gain
  • Unusual tiredness

Heart Rate Changes. Betaxolol can make your heart beat slower than normal (bradycardia). Call your healthcare provider right away if you have any of the following symptoms of bradycardia. 

  • Feeling lightheaded, dizziness, or fainting
  • Confusion
  • Feeling weak or easily tired 
  • Chest pain
  • Shortness of breath

Decreased Blood Pressure (Hypotension). Betaxolol may cause low blood pressure. If you feel faint or dizzy, lie down. Tell your healthcare provider right away if you have any of the following symptoms of low blood pressure.

  • Dizziness, feeling lightheaded, or fainting
  • Confusion
  • Feeling weak or tired

Breathing Problems. Betaxolol may cause the muscles around the airways to tighten (bronchospasm) instead of relaxing, which can be serious. Stop using betaxolol and contact your healthcare provider right away if you have trouble breathing.

Severe Allergic Reactions. Betaxolol may cause allergic reactions, which can be serious. Stop using betaxolol and get help right away if you have any of the following symptoms of a serious allergic reaction.

  • Breathing problems or wheezing
  • Racing heart
  • Fever or general ill feeling
  • Swollen lymph nodes
  • Swelling of the face, lips, mouth, tongue, or throat
  • Trouble swallowing or throat tightness
  • Itching, skin rash, or pale red bumps on the skin called hives
  • Nausea or vomiting
  • Dizziness, feeling lightheaded, or fainting
  • Stomach cramps
  • Joint pain

Warnings & Precautions

Who should not use betaxolol?

Allergies to Ingredients. People who are allergic to any of the following should not use betaxolol.

  • Kerlone
  • Betaxolol
  • Any of the ingredients in the specific product dispensed

Your pharmacist can tell you all of the ingredients in the specific betaxolol products they stock.

Bradycardia. Betaxolol should not be used if your heart is beating too slow (bradycardia).

Heart Block. Betaxolol should not be used if the electrical signals in your heart move too slow (heart block).

Severe or Worsening Heart Failure. Betaxolol should not be used if your heart failure is severe or getting worse, causing you to feel very tired, have trouble breathing, or swelling in your legs. 

Cardiogenic Shock. Betaxolol should not be used if you have a life-threatening condition called cardiogenic shock where your heart cannot pump enough blood to the rest of your body.

Untreated Pheochromocytoma. Betaxolol should not be used in people with a certain type of adrenal gland tumor, called pheochromocytoma, if it is not being treated. 

What should I know about betaxolol before using it?

Do not take betaxolol unless it has been prescribed to you by a healthcare provider. Take it as prescribed.

Do not share betaxolol with other people, even if they have the same condition as you. It may harm them.

Keep betaxolol out of the reach of children.

Betaxolol can affect your alertness or coordination. Do not drive or do other activities that require alertness or coordination until you know how betaxolol affects you.

Stopping betaxolol suddenly may lead to chest pain and heart attack in people with heart disease. Do not stop taking this medication without talking to your healthcare provider first. 

What should I tell my healthcare provider before using betaxolol?

Tell your healthcare provider about all of your health conditions and any prescription or over-the-counter (OTC) medicines, vitamins/minerals, herbal products, and other supplements you are using. This will help them determine if betaxolol is right for you.

In particular, make sure that you discuss any of the following.

Current and Past Health Conditions. Tell your healthcare provider if you have any of the following.

  • Heart problems
  • Breathing problems
  • Kidney problems
  • Thyroid problems

Diabetes. Betaxolol can decrease early signs of low blood sugar, such as fast heartbeat, and make it more likely for the low blood sugar to be serious, especially for people with diabetes.

Pregnancy. It is not known if or how betaxolol could affect pregnancy or harm an unborn baby. Tell your healthcare provider if you are or plan to become pregnant.

Breastfeeding. Betaxolol passes into breast milk. Tell your healthcare provider if you are breastfeeding or plan to breastfeed.

Interactions

Does betaxolol interact with foods or drinks?

There are no known interactions between betaxolol and foods or drinks.

It is unknown if drinking alcohol will affect betaxolol. The risk of dizziness may be increased if you drink alcohol while taking betaxolol.

Does betaxolol interact with other medicines (drug interactions)?

Always tell your healthcare provider about any prescription or over-the-counter (OTC) medicines, vitamins/minerals, herbal products, and other supplements you are using.

In particular, make sure that you discuss if you are using any of the following before taking betaxolol.

  • Diltiazem and verapamil, which are medicines used to treat chest pain and high blood pressure
  • Digoxin (Lanoxin), which is a medicine used to treat irregular heartbeat and some types of heart failure
  • Clonidine, which is a medicine used to treat high blood pressure and attention deficit hyperactivity disorder (ADHD)
  • Any medicine for irregular heart rate or rhythm
  • Any medicine for high blood pressure 
  • Any medicine for diabetes
Does Betaxolol interact with other drugs you are taking?
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Overdose/Missed Dose

What should I do if I accidentally use too much betaxolol?

If you or someone else has used too much betaxolol, get medical help right away, call 911, or contact a Poison Control center at 800-222-1222.

What should I do if I miss a dose of betaxolol?

If you miss a dose, take it as soon as you remember. If it is almost time for your next dose, skip the missed dose and only take the next dose. Do not take double or extra doses.

Drug Survey

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